Keywords: GPCR activation.png en Schematic representation of the two state-model of CB1 receptor activation in which receptors are in equilibrium between two states active and inactive R and R An agonist will stabilize the active state leading to activation a neutral antagonist binds equally to active and inactive states whereas an inverse agonist will preferentially stabilize the inactive state My own work Created in Microsoft Word Dagrun Saevarsdottir 2008-11-12 - Medicinal chemistry G protein coupled receptors |